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PROTEASOME INHIBITOR

外国特許コード F130007461
掲載日 2013年7月4日
出願国 世界知的所有権機関(WIPO)
国際出願番号 2012JP065992
国際公開番号 WO 2012/176878
国際出願日 平成24年6月22日(2012.6.22)
国際公開日 平成24年12月27日(2012.12.27)
優先権データ
  • 特願2011-139235 (2011.6.23) JP
発明の名称 (英語) PROTEASOME INHIBITOR
発明の概要(英語)

[Problem] To provide a novel proteasome inhibitor which can be administered orally. [Solution] A proteasome inhibitor comprising, as an active ingredient, a compound represented by general formula (1) [wherein Y and Y' are the same as or different from each other and independently represent a single bond, -O-, -NH-, -CH=CH?, -CO-CH=CH?, -O-CONH?, -S-CO?, -CONH?, -NHCO? or NHSO2? [wherein "?" represents a bond located on the phenyl group side]

R1, R2, R3, R4, R5, R6, R7 and R8 are the same as or different from one another and independently represent a hydrogen atom, a halogen atom, a hydroxy group, an amino group, a carboxyl group, a C1-6 alkyl group, a C1-6 alkoxy group or a C1-6 alkoxycarbonyl group

R9 and R10 are the same as or different from each other and independently represent a hydrogen atom or a C1-6 alkyl group, or R9 and R10 together form -CH2CH2- or -CH2CH(R11)CH2- [wherein R11 represents a hydrogen atom, a C1-6 alkoxy group or a C1-6 alkylsulfonyloxy group]

and m and n are the same as or different from each other and independently represent an integer of 2-4] or a salt thereof, or a solvate of the compound or the salt.

  • 出願人(英語)
  • ※2012年7月以前掲載分については米国以外のすべての指定国
  • EDUCATIONAL FOUNDATION JICHI MEDICAL UNIVERSITY,
  • KOWA COMPANY, LTD,
  • FURUKAWA, YUSUKE,
  • KIKUCHI, JIRO
  • 発明者(英語)
  • FURUKAWA, YUSUKE,
  • KIKUCHI, JIRO
国際特許分類(IPC)
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