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PDK4 INHIBITOR AND USE THEREOF

外国特許コード F140008051
整理番号 S2013-0371-C0
掲載日 2014年12月4日
出願国 世界知的所有権機関(WIPO)
国際出願番号 2013JP007649
国際公開番号 WO 2014103321
国際出願日 平成25年12月26日(2013.12.26)
国際公開日 平成26年7月3日(2014.7.3)
優先権データ
  • 61/745,819P (2012.12.26) US
発明の名称 (英語) PDK4 INHIBITOR AND USE THEREOF
発明の概要(英語) [Problem] The problem of the present invention is to provide a novel pyruvate dehydrogenase inhibitor. [Solution] Provided are a pyruvate dehydrogenase inhibitor comprising the compound represented by general formula (I) as the active ingredient (where in the formula, ring A is a six-member hydrocarbon ring having aromaticity that is optionally substituted by two to four substitution groups, R1 and R4 are the same or different and are, for instance, a hydrogen atom, hydroxyl group, or optionally substituted C1-6 alkyl group, and R2 and R3 are the same or different and are a hydrogen atom, carboxyl group, optionally substituted C1-6 alkyl group, C6-10 aryl group, or -C(=R9)-R10); a medical composition which comprises the pyruvate dehydrogenase kinase inhibitor as the active ingredient and which is for treating or preventing a disease or an impairment the development or deterioration of which is associated with pyruvate dehydrogenase kinase; and a cosmetic composition, and the like.
  • 出願人(英語)
  • ※2012年7月以前掲載分については米国以外のすべての指定国
  • THE KITASATO INSTITUTE
  • UNIVERSITY OF TOKUSHIMA
  • 発明者(英語)
  • OMURA SATOSHI
  • NAKANO HIROFUMI
  • YAMAJI KENZABURO
  • YAMAMOTO TSUYOSHI
  • KIDO HIROSHI
  • YAMANE KAZUHIKO
  • SUNAZUKA TOSHIAKI
  • HIROSE TOMOYASU
国際特許分類(IPC)
指定国 National States: AE AG AL AM AO AT AU AZ BA BB BG BH BN BR BW BY BZ CA CH CL CN CO CR CU CZ DE DK DM DO DZ EC EE EG ES FI GB GD GE GH GM GT HN HR HU ID IL IN IR IS JP KE KG KN KP KR KZ LA LC LK LR LS LT LU LY MA MD ME MG MK MN MW MX MY MZ NA NG NI NO NZ OM PA PE PG PH PL PT QA RO RS RU RW SA SC SD SE SG SK SL SM ST SV SY TH TJ TM TN TR TT TZ UA UG US UZ VC VN ZA ZM ZW
ARIPO: BW GH GM KE LR LS MW MZ NA RW SD SL SZ TZ UG ZM ZW
EAPO: AM AZ BY KG KZ RU TJ TM
EPO: AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
OAPI: BF BJ CF CG CI CM GA GN GQ GW KM ML MR NE SN TD TG

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