TOP > 外国特許検索 > ANTI-GRAM-NEGATIVE-BACTERIA AGENT, THERAPEUTIC AND PROPHYLACTIC AGENT AGAINST GRAM-NEGATIVE BACTERIAL INFECTIONS CONTAINING SAME, AND DISINFECTANT AGAINST GRAM-NEGATIVE BACTERIA

ANTI-GRAM-NEGATIVE-BACTERIA AGENT, THERAPEUTIC AND PROPHYLACTIC AGENT AGAINST GRAM-NEGATIVE BACTERIAL INFECTIONS CONTAINING SAME, AND DISINFECTANT AGAINST GRAM-NEGATIVE BACTERIA

外国特許コード F160008901
整理番号 (S2015-0858-N0)
掲載日 2016年11月11日
出願国 世界知的所有権機関(WIPO)
国際出願番号 2016JP058659
国際公開番号 WO 2016152764
国際出願日 平成28年3月18日(2016.3.18)
国際公開日 平成28年9月29日(2016.9.29)
優先権データ
  • 特願2015-058273 (2015.3.20) JP
発明の名称 (英語) ANTI-GRAM-NEGATIVE-BACTERIA AGENT, THERAPEUTIC AND PROPHYLACTIC AGENT AGAINST GRAM-NEGATIVE BACTERIAL INFECTIONS CONTAINING SAME, AND DISINFECTANT AGAINST GRAM-NEGATIVE BACTERIA
発明の概要(英語) The problem to be solved by the present invention is to provide a low-molecular compound that demonstrates an antibacterial effect against gram-negative bacteria, and particularly against multidrug-resistant gram-negative bacteria, even when used alone, without combination with other agents. This anti-gram-negative bacteria agent is characterized by comprising a compound represented by formula (I) (R11, R12, R13, R14, R15, R21, R22, R23, R24, R25 and R31 each individually represent a hydrogen atom or a predetermined substituent).
特許請求の範囲(英語) [claim1]
1. The chemical compound which is displayed with formula (i) or it features that salt is contained, the anti- gram negative germ medicine.
In formula (i), R (11), R (12), R (13), R (14), R (15), R (21), R (22), R (23), R (24), R (25) and R (31) respectively becoming independent, the hydrogen atom and the halogen atom, the number of carbon atoms the 1-4 the alkyl group (- R), the hydroxyl basis (- OH), the number of carbon atoms the 1-4 alkoxy group (- OR), the [merukaputo] basis (- SH), the number of carbon atoms the 1-4 thio alkoxy group (-SR) The carboxyl group (- COOH), the number of carbon atoms the 2-5 the carboxylic acid ester basis (- COO-R), is connected to the nitrogen atom of end the hydrogen atom which the number of carbon atoms the 1-4 may be substituted with the alkyl group the carboxylic acid amide basis (- COO-NH [2]), the number of carbon atoms the 2-5 the acyl basis (- CO-R), is connected to the nitrogen atom of end the hydrogen atom which the number of carbon atoms the 1-4 may be substituted with the alkyl group the [karubamoiru] basis (- CO-NH [2]), is connected to the nitrogen atom the hydrogen atom which the number of carbon atomsThe amino group the 1-4 may be substituted with the alkyl group (- NH [2]), the hydrogen atom which is connected to the nitrogen atom of end the number of carbon atoms the [ureido] basis the 1-4 may be substituted with the alkyl group (- NH-CO-NH [2]), the nitro group (- NO [2]) or the cyano basis (- CN) you display.
[claim2]
2. At least one of the following conditions is satisfied, in claim 1 the anti- gram negative germ medicine of statement:
(i) R (11), R (12), R (13), R (14) or R (15), the number of carbon atoms the 1-4 it is the alkyl group;
(ii) R (23), the hydrogen atom, the number of carbon atoms the 1-4 the alkyl group and the hydroxyl basis, the number of carbon atoms the hydrogen atom which the 1-4 connects to thio alkoxy group, or the nitrogen atom the number of carbon atoms is the amino group the 1-4 may be substituted with the alkyl group;
(iii) R (31) is the hydrogen atom;
(iv) R (11), R (12), R (13), R (14) and R (15) the quantity of those which are the substituent inside and other than the hydrogen atom is 2 or less;
(v) R (21), R (22), R (23), R (24) and R (25) the quantity of those which are the substituent inside and other than the hydrogen atom is 2 or less.
[claim3]
3. The chemical compound which is displayed with aforementioned formula (i), the chemical compound of 10 types which are displayed with the below-mentioned formula: It is either A-1-A-4 and C-1-C-6, in claim 1 or 2 the anti- gram negative germ medicine of statement.
[claim4]
4. The medicine tolerance gram negative germ is dealt with of application, either of the claim 1-3 in one section the anti- gram negative germ medicine of statement.
[claim5]
5. The aforementioned medicine tolerance gram negative germ is the multi medicine tolerance green pus germs or the multi medicine tolerance [ashinetobakuta] being attached germs, in claim 4 the anti- gram negative germ medicine of statement.
[claim6]
6. Either of the claim 1-5 it features that it contains the anti- gram negative germ medicine of statement in one section as the active ingredient, the remedy or the preventive medicine for the gram negative germ infection symptom.
[claim7]
7. Either of the claim 1-5 it features that it contains the anti- gram negative germ medicine of statement in one section as the active ingredient, the disinfectant for the gram negative germ.
  • 出願人(英語)
  • ※2012年7月以前掲載分については米国以外のすべての指定国
  • TOKAI UNIVERSITY EDUCATIONAL SYSTEM
  • 発明者(英語)
  • YOSHIHARA EISAKU
国際特許分類(IPC)
指定国 National States: AE AG AL AM AO AT AU AZ BA BB BG BH BN BR BW BY BZ CA CH CL CN CO CR CU CZ DE DK DM DO DZ EC EE EG ES FI GB GD GE GH GM GT HN HR HU ID IL IN IR IS JP KE KG KN KP KR KZ LA LC LK LR LS LU LY MA MD ME MG MK MN MW MX MY MZ NA NG NI NO NZ OM PA PE PG PH PL PT QA RO RS RU RW SA SC SD SE SG SK SL SM ST SV SY TH TJ TM TN TR TT TZ UA UG US UZ VC VN ZA ZM ZW
ARIPO: BW GH GM KE LR LS MW MZ NA RW SD SL SZ TZ UG ZM ZW
EAPO: AM AZ BY KG KZ RU TJ TM
EPO: AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
OAPI: BF BJ CF CG CI CM GA GN GQ GW KM ML MR NE SN ST TD TG
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